Bioactivity:Peptide fragment containing amino acids 1-11 of Nociceptin. Potent agonist of the ORL1/KOR-3 receptor (Ki = 55 nM); displays no affinity for opioid receptors, including μ, δ, κ1 and κ3 receptors (Ki >1000 nM). Displays analgesic properties in CD-1 mice.
CAS Nr:
178249-41-7
Purity:
98%
SMILES:
Formula:
C49H75N15O14
Molecular weight:
1098,2
Pathway:
Target: